Search results for "Sodium channel"

showing 10 items of 50 documents

Novel mutations in the voltage-gated sodium channel of pyrethroid-resistant Varroa destructor populations from the Southeastern USA

2016

The parasitic mite Varroa destructor has a significant worldwide impact on bee colony health. In the absence of control measures, parasitized colonies invariably collapse within 3 years. The synthetic pyrethroids tau-fluvalinate and flumethrin have proven very effective at managing this mite within apiaries, but intensive control programs based mainly on one active ingredient have led to many reports of pyrethroid resistance. In Europe, a modification of leucine to valine at position 925 (L925V) of the V. destructor voltage-gated sodium channel was correlated with resistance, the mutation being found at high frequency exclusively in hives with a recent history of pyrethroid treatment. Here,…

0106 biological sciences0301 basic medicineInsecticidesVeterinary medicineGene Identification and Analysislcsh:MedicineMicrobiologiaVoltage-Gated Sodium ChannelsFlumethrinmedicine.disease_causeBiochemistry01 natural sciencesAbellesInsecticide Resistancechemistry.chemical_compoundMethioninePyrethrinsÀcarsDestructorAmino Acidslcsh:ScienceMitesMutationMultidisciplinaryPyrethroidbiologyOrganic CompoundsGeneral MedicineBeesSoutheastern United StatesInsectsChemistryPhysical SciencesInsect ProteinsGeneral Agricultural and Biological SciencesResearch ArticleArthropodaApiaryParàsitsVarroidaeGeneral Biochemistry Genetics and Molecular Biology03 medical and health sciencesLeucineparasitic diseasesGeneticsMitemedicineAnimalsPoint MutationSulfur Containing Amino AcidsIsoleucineMutation DetectionAllelesbusiness.industryPoint mutationOrganic Chemistrylcsh:ROrganismsChemical CompoundsBiology and Life SciencesProteinsbiology.organism_classificationInvertebratesHymenopteraBiotechnology010602 entomology030104 developmental biologyAliphatic Amino AcidschemistryGenetic LociVarroa destructorMutationlcsh:Qbusiness
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Mutations in the voltage-gated sodium channel gene associated with deltamethrin resistance in commercially sourced Phytoseiulus persimilis

2020

The implementation of Integrated Pest Management (IPM) in current agricultural practice is a convenient and very effective strategy to maintain pest populations under control. The use of Biological Control Agents, like Phytoseiulus persimilis, is key for the success of such approach. This predatory mite is widely used since it is very effective for controlling the two spotted spider mite (Tetranychus urticae), one of the most devastating pests worldwide. Here we show the identification of mutations located in the Voltage Gated Sodium Channel (VGSC) of P. persimilis, that correlate with the reduced susceptibility to deltamethrin observed in commercially sourced colonies of this predatory mit…

0106 biological sciences0301 basic medicineIntegrated pest managementPyrethroid resistancePhytoseiulus persimilisVoltage gated sodium channelDrug ResistanceBiological pest controlVoltage-Gated Sodium Channels01 natural sciencesArthropod ProteinsToxicology03 medical and health scienceschemistry.chemical_compoundPlagues ControlSpider miteNitrilesPyrethrinsparasitic diseasesPlaguicidesGeneticsMiteAnimalsPoint MutationÀcarsAmino Acid SequenceTetranychus urticaeMolecular BiologyAcaricidesBase SequencebiologyPesticidebiology.organism_classification010602 entomology030104 developmental biologyDeltamethrinchemistryInsect ScienceMutationPEST analysisTetranychidaeSequence Alignment
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Mutations in voltage-gated sodium channels from pyrethroid resistant salmon lice (Lepeophtheirus salmonis)

2018

BACKGROUND Parasitic salmon lice (Lepeophtheirus salmonis) cause high economic losses in Atlantic salmon farming. Pyrethroids, which block arthropod voltage-gated sodium channels (Nav 1), are used for salmon delousing. However, pyrethroid resistance is common in L. salmonis. The present study characterized Nav 1 homologues in L. salmonis in order to identify channel mutations associated to resistance, called kdr (knockdown) mutations. RESULTS Genome scans identified three L. salmonis Nav 1 homologues, LsNav 1.1, LsNav 1.2 and LsNav 1.3. Arthropod kdr mutations map to specific Nav 1 regions within domains DI-III, namely segments S5 and S6 and the linker helix connecting S4 and S5. The above …

0106 biological sciencesGeneticsMutationGene knockdownPyrethroidbiologySodium channelGeneral Medicinebiology.organism_classificationmedicine.disease_cause01 natural sciencesGenome010602 entomologychemistry.chemical_compoundDeltamethrinchemistryLepeophtheirusInsect Scienceparasitic diseasesmedicineAgronomy and Crop ScienceAllele frequency010606 plant biology & botanyPest Management Science
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Mutations associated with pyrethroid resistance in Varroa mite, a parasite of honey bees, are widespread across the United States.

2021

BACKGROUND Managed honey bees are key pollinators of many crops and play an essential role in the United States food production. For more than ten years, beekeepers in the United States have been reporting high rates of colony losses. One of the drivers of these losses is the parasitic mite Varroa destructor. Maintaining healthy honey bee colonies in the United States is dependent on a successful control of this mite. The pyrethroid tau-fluvalinate (Apistan®) was among the first synthetic varroacides registered in the United States. With over 20 years of use, mites resistant to Apistan® have emerged, and so it is unsurprising that treatment failures have been reported. Resistance to tau-flu…

0106 biological sciencesIntegrated pest managementApiaryVarroidaeVoltage-Gated Sodium Channels01 natural sciencesparasitic diseasesPyrethrinsMiteAnimalsParasitesbiologybusiness.industryKnockdown resistanceGeneral MedicineHoney beeBeesbiology.organism_classificationUnited StatesBiotechnology010602 entomologyInsect ScienceVarroa destructorMutationVarroaPEST analysisbusinessAgronomy and Crop Science010606 plant biology & botanyPest management scienceReferences
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Investigation of deltamethrin resistance in salmon lice (Lepeophtheirus salmonis) provides no evidence for roles of mutations in voltage-gated sodium…

2020

BACKGROUND The pyrethroid deltamethrin is used to treat infestations of farmed salmon by parasitic salmon lice, Lepeophtheirus salmonis (Kroyer). However, the efficacy of deltamethrin for salmon delousing is threatened by resistance development. In terrestrial arthropods, knockdown resistance (kdr) mutations of the voltage-gated sodium channel (Nav ), the molecular target for pyrethroids, can cause deltamethrin resistance. A putative kdr mutation of an L. salmonis sodium channel homologue (LsNav 1.3 I936V) has been identified previously. At the same time, deltamethrin resistance of L. salmonis has been shown to be inherited maternally and to be associated with mitochondrial DNA (mtDNA) muta…

0106 biological sciencesMaleMitochondrial DNALocus (genetics)Voltage-Gated Sodium ChannelsBiology01 natural sciencesCopepodaInsecticide Resistancechemistry.chemical_compoundFish DiseasesEtofenproxSalmonparasitic diseasesGenotypeNitrilesPyrethrinsAnimalsGeneticsPyrethroidKnockdown resistanceGeneral Medicinebiology.organism_classification010602 entomologyDeltamethrinchemistryLepeophtheirusInsect ScienceMutationFemaleAgronomy and Crop Science010606 plant biology & botanyPest management scienceREFERENCES
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Dendritic and Axonal L-Type Calcium Channels Cooperate to Enhance Motoneuron Firing Output during Drosophila Larval Locomotion

2017

Behaviorally adequate neuronal firing patterns are critically dependent on the specific types of ion channel expressed and on their subcellular localization. This study combinesin situelectrophysiology with genetic and pharmacological intervention in larvalDrosophila melanogasterof both sexes to address localization and function of L-type like calcium channels in motoneurons. We demonstrate that Dmca1D (Cav1 homolog) L-type like calcium channels localize to both the somatodendritic and the axonal compartment of larval crawling motoneurons.In situpatch-clamp recordings in genetic mosaics reveal that Dmca1D channels increase burst duration and maximum intraburst firing frequencies during craw…

0301 basic medicineBK channelSodium ChannelsSK channel03 medical and health sciences0302 clinical medicineAnimalsDrosophila ProteinsLarge-Conductance Calcium-Activated Potassium ChannelsResearch ArticlesMotor NeuronsVoltage-dependent calcium channelbiologyGeneral NeuroscienceSodium channelCalcium channelfungiExcitatory Postsynaptic PotentialsAfterhyperpolarizationDendritic CellsAxonsElectrophysiological PhenomenaElectrophysiologyStretch-activated ion channel030104 developmental biologyDrosophila melanogasternervous systemLarvaSynapsesbiology.proteinCalcium ChannelsNeuroscience030217 neurology & neurosurgeryLocomotion
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Prognostic Challenges of SCN1A Genetic Mutations: Report on Two Children with Mild Features

2016

Mutations in the gene encoding the α-1 subunit of the voltage-gated sodium channel (SCN1A) are associated with variable but usually severe clinical course, both for the epileptic seizures and the cognitive impairment. The purpose of the present study was to retrospectively review two patients affected by seizures and two different types of SCN1A gene mutations (microdeletion and point mutation). The children (a 4-year-old girl and a 3-year-old boy) were affected by generalized tonic–clonic seizures and myoclonic jerks plus unilateral seizures, respectively. Genetic analyses showed, in the girl, the presence of a 4 MB deletion involving SCN1A and four other genes, and a point mutation in the…

0301 basic medicinePediatricsmedicine.medical_specialtybusiness.industryPoint mutationmedia_common.quotation_subjectSodium channel geneMyoclonic JerkClinical course030105 genetics & hereditymedicine.disease03 medical and health sciences0302 clinical medicineDravet syndromePediatrics Perinatology and Child HealthGenotypemedicineNeurology (clinical)GirlbusinessGene030217 neurology & neurosurgerymedia_commonJournal of Pediatric Neurology
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Human CD8(+) T Cells Damage Noninfected Epithelial Cells during Influenza Virus Infection In Vitro

2017

During severe influenza A virus (IAV) infections, a large amount of damage to the pulmonary epithelium is the result of the antiviral immune response. Specifically, whilst CD8+ T cells are important for killing IAV-infected cells, during a severe IAV infection, they can damage uninfected epithelial cells. At present, the mechanisms by which this occurs are unclear. Here, we used a novel in vitro coculture model of human NCl-H441 cells and CD8+ T cells to provide a new insight into how CD8+ T cells may affect uninfected epithelial cells during severe IAV infections. Using this model, we show that human IAV-specific CD8+ T cells produce soluble factors that reduce the barrier integrity of non…

0301 basic medicinePulmonary and Respiratory MedicineEpithelial sodium channelCD8(+) T cellsClinical BiochemistryCell BiologyLung injuryBiologyVirologyinfluenza virusepithelial cellsbystander damage03 medical and health sciencesInterleukin 21030104 developmental biology0302 clinical medicineImmune systemBystander effectCytotoxic T cellTumor necrosis factor alphaMolecular BiologyCD8030215 immunologyAmerican Journal of Respiratory Cell and Molecular Biology
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Extracellular electrical recording of pH-triggered bursts in C6 glioma cell populations

2016

Extracellular electrode recording demonstrates acid-triggered electrical activity in glioma cell populations.

0301 basic medicinegliaAcid-sensing ion channelsbioelectronicsBiologySodium Channels03 medical and health sciencesBurstingchemistry.chemical_compound0302 clinical medicineCell Line TumorGliomaASICsPsalmotoxinmedicineExtracellularAnimalsHumansneoplasmsResearch ArticlesAcid-sensing ion channelIon channelLow frequency current noiseNeuronsBioelectronicsMultidisciplinarySodium channelSciAdv r-articlesGliomaHydrogen-Ion Concentrationmedicine.diseaseC6 Gliomanervous system diseasesElectrophysiological PhenomenaRatsPcTX-1030104 developmental biologychemistryCell cultureBiophysicsASICs; Acid-sensing ion channels; C6 Glioma; Electrical recording; Low frequency current noise; PcTX-1; bioelectronics; gliaNerve Net030217 neurology & neurosurgeryResearch ArticleElectrical recordingScience Advances
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Sustained seizure freedom with adjunctive brivaracetam in patients with focal onset seizures

2022

The maintenance of seizure control over time is a clinical priority in patients with epilepsy. The aim of this study was to assess the sustained seizure frequency reduction with adjunctive brivaracetam (BRV) in real-world practice. Patients with focal epilepsy prescribed add-on BRV were identified. Study outcomes included sustained seizure freedom and sustained seizure response, defined as a 100% and a ≥50% reduction in baseline seizure frequency that continued without interruption and without BRV withdrawal through the 12-month follow-up. Nine hundred ninety-four patients with a median age of 45 (interquartile range = 32-56) years were included. During the 1-year study period, sustained se…

AdultFreedomfocal seizuresEpilepsiesSettore MED/26Double-Blind MethodDrug Therapyantiseizure medication; brivaracetam; focal seizures; seizure freedom; sodium channel blockers; Adult; Double-Blind Method; Drug Therapy Combination; Freedom; Humans; Middle Aged; Pyrrolidinones; Seizures; Treatment Outcome; Anticonvulsants; Epilepsies PartialSeizuresseizure freedomHumansanti-seizure medication; focal seizures; epilepsyantiseizure medicationbrivaracetamanti-seizure medicationMiddle AgedPyrrolidinonesTreatment OutcomeNeurologysodium channel blockersCombinationepilepsyDrug Therapy CombinationAnticonvulsantsNeurology (clinical)Epilepsies PartialPartial
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